Target (protein): Type II site-specific deoxyribonuclease
E.C Number: 3.1.21.4
Protein ID: WP_000781649.1
PDB ID: 1STX
Organism: Escherichia coli
Etiologic Risk Group (see link below): N/a
Disease Information:
Escherichia Coli are bacteria that live in the intestines and are usually harmless but some of them can be pathogenic. They can cause diarrhea or infection outside of the intestinal tract. These types of bacteria are transmitted through contaminated water, food, or contact with another person or animal. The six types of E.Coli that cause this disease are Shiga toxin producing E.coli (STEC), Enterotoxigenic E. coli (ETEC), Enteropathogenic E. coli (EPEC), Enteroaggregative E. coli (EAEC), Enteroinvasive E. coli (EIEC) and Diffusely adherent E. coli (DAEC). Unfortunately, there is not a cure for E.Coli infections, it has to run its course and eventually get out of the body. To prevent from contracting en E.Coli infection maintain hands clean, cook meat thoroughly, wash vegetables, store foods separately, and get pasteurized drinks.
Links:
  1. http://www.medicalnewstoday.com/articles/68511.php
  2. https://www.cdc.gov/ecoli/general/index.html
  3. https://www.patricbrc.org/view/Feature/RefSeq.356829.3.JGZU01000001.CDS.4223.5182.fw

Link to TDR Targets page (if present): N/A

Essentiality of Type II site-specific deoxyribonuclease:
The Type II site-specific deoxyribonuclease is an enzyme that helps catalyze endonucleolytic cleavage of DNA to give specific double-stranded fragments with terminal 5'-phosphates.
Links:
  1. http://enzyme.expasy.org/EC/3.1.21.4


Druggable Target: Not available


Link to BRENDA: http://www.brenda-enzymes.org/enzyme.php?ecno=3.1.21.4

Enzyme Assay Information: http://www.sciencedirect.com/science/article/pii/S002228360301297X

Eco RV assay of DNA using N6-methyladenine

http://www.sigmaaldrich.com/catalog/product/roche/ecorvro?lang=en&region=US&cm_sp=Insite-_-prodRecCold_xviews-_-prodRecCold10-1

Reagents and Materials:
Relative activity in PCR mix (Taq DNA Polymerase buffer) is 10%. The PCR mix contained λDNA, primers, 10 mM Tris-HCl (pH 8.3, 20 °C), 50 mM KCl, 1.5 mM MgCl2, 200 μM dNTPs, 2.5 U Taq DNA polymerase. The mix was subjected to 25 amplification cycles. Activity in reaction buffer of Pwo SuperYield DNA Polymerase PCR Mix is 25%. When supplemented with GC-RICH Solution activity remains at 25%.
The Eco RV assay that contains all of these materials in it is worth $62.


Structure (PDB)
Sequence ID: WP_000781649.1

Show pairwise alignment of your BLASTP search in NCBI:


Capture.PNG
Query Coverage: 100%
Max % Identities: 100%
% Positives: 100%
Chain used for homology: A


Inhibitors: EDTA

Expression Information:
The target has been expressed in E.Coli. It is expressed predominatley in bacteria because it is a restriction modification system that helps protect the bacteria from foreign DNA that tries to inhibit it.
Link:
  1. https://www.ncbi.nlm.nih.gov/pubmed/10510229

Purification Method: Heparin-Sepharose column chromatography

Image of Protein:
Capture 2.PNG

Figure 1: Structure of the K38A mutant of EcoRV bound to cognate DNA and Mn2

*Amino Acid Sequence (paste as text only - not as screenshot or as 'code'):
<span style="background-color: #ffffff; color: #626262;">  1__0__         2__0__         3__0__         4__0__         5__0__         6__0__
MNNQNDYIEA AQQIIASLGL PRAQQNERSA LCLLALLNLT PGKAWADAEN PLVGITPIMN
 
        7__0__         8__0__         9__0__        10__0__        11__0__        12__0__
WVREHYGKVY APNTRETFRR QSMHQFCAAG VALYNPDKPD RPVNSPKAVY QIEPAALSML
 
       13__0__        14__0__        15__0__        16__0__        17__0__        18__0__
RTFGSPAWHD SLATYLAERE TLVTRYAKER EQNRIPVEIA AGQQITLSPG EHSELIRAII
 
       19__0__        20__0__        21__0__        22__0__        23__0__        24__0__
EDFAPRFAPG SVLVYAGDTG EKWGYFDAPL LAGLGVDVDS HGKMPDVVLH FTAKNWLLLV
 
       25__0__        26__0__        27__0__        28__0__        29__0__        30__0__
ESVTSHGPVD GKRHAELARL FAGSTAGLVY VTAFPNRSIM GRYLGEIAWE TEVWVADAPS
 
       31__0__
HLIHFNGVRF LGPYSTE </span>
*length of your protein in Amino Acids: 317
Molecular Weight of your protein in kiloDaltons using the Expasy ProtParam website: 35064.82 KDa
Molar Extinction coefficient of your protein at 280 nm wavelength: 56505
TMpred graph Image (http://www.ch.embnet.org/software/TMPRED_form.html). Input your amino acid sequence to it.



Capture 3.PNG
Figure 2: TMPred output graph for Type II site-specific deoxyribonuclease
*CDS Gene Sequence (paste as text only):
<span style="background-color: #ffffff; font-family: monospace,serif;">NC_017527.1:757901-761041 Methanosaeta harundinacea 6Ac, complete genome
<span class="ff_line">GTGGCCGTTCCGGAGAAGATCCTTGAGTTGGTTGAAAAATTCGAATTGGTCATTGATAAATATAAATCTA
GTTATAAAGAAGAAGAAATTAAAATTGAATTTATAAATCCTTTTTTTGAAGCTCTAGGCTGGGATGTCCG
AAATAAGAGCAATAACCCCCCAGATCAGAGAGAGGTCAGGTTTGAAGATACCTTGAGGTCAGAGGGGGAG
ACCCAGAGGCCCGATTATAGCTTCTGGCTTGACAGGGAGAGGAAGTTCTTTCTGGACGCCAAAAAACCTT
CAGTGAATATTGAAGGAGGAATAATCCCAGCATTCCAGATAAAGCGTTATGCATACTCTTCTACCCTGCC
GCTTGCCATTGTAACCGACTTTGAAGAGTTTGCCGTTTACGATTGCAGGATCAAACCGTTCAAATTTGAT
AAGCCACAAAAGTCTAGATTATTATTAATAAAATATTATGAATATGAAAAGAGATGGGACGAGATCGCCT
CGTTGTTCTCCAAAGAGGCCGTTCAGAGAGGCTCCCTCGGCTCCATCCCTCCGCCAAAAGGAAAAAAAGT
CGACGACGCTCTTCTGGAGGACATCTCTGATTGGCGAAATGCTCTGGCGGCGAGCATCACTAAGATGAAT
CCAGAGATCTCTCAGAAGAGCCTGAACTATGCGGTCCAGATGACGATCGACAGGATTCTATTTCTAAGGA
TCTGTGAGGATCGGTCTATTGAGGACAGCGAGCGGTTGAAGGGGCTTCTTGATGGGGATGATGTATATAA
GAGGCTGTTTGAACTCTTCGAAGAGGCCGATAAGAGGTACAATTCGGGGCTGTTCCACTTCCATCCTGAG
GAGGAGAGGAACAACTTCGACGCCATCACCCCGTCGATAAAGATCGAGGACAATGTTCTTAAGAATATAA
TTCAAAGCTTATACTATCCTGACAGCCCCTACGTCTTCTCTGAGATCCCTGCCGATATTCTTGGTCACGT
TTACGAGCAGTTCCTGGGGAAGGTCATCCAGCTGGACGAGAGCCACAAAGTGAGCGTGGTGGAGAAGCCT
GAGGTGAGGAAGGCAGGAGGCGTTTATTATACTCCATCATATATTGTAGATTATATCGTTAAAAACACCG
TCGGCAAGCTCTTGGAGGGGAAGACCCCCAAGGAGGCCTCTGACCTTCGCATCCTCGATCCCGCCTGCGG
TTCGGGGTCGTTTCTGATAGTGGCCTATCAGCACCTCTTGGATTGGCACCTCGACTGGTACAAGGCCCAT
CTCGTCCCTCTCTTGGATGCTGGAGAGAAGCCGACATCAAACGGGGTGCAAAATCTCCTCCCGTCTCCGA
TCGAGAGGCCAGGGAAGAACGCCAGGTCCCGATCGAAGAAGATCTGGGAGAGGGCTTCGGTGGCGACCCT
CCCCATCGAGGAGAGGGCGGGAGAATGGCATCTGAAGACCGCCGAGAGGAAGAGGATCCTCCTCAACAAC
ATCTATGGCGTGGATATAGACACTCAGGCCGTGGAGGTGACAAAGCTCTCCCTCCTCCTCAAGGTCTTGG
AAGGAGAAAATAAGGCCACCATCACCGATCTCAACATGTATTCAGATGAGAGGGCTCTGCCAGATCTTGG
AAATAATATAAAATGTGGCAATTCCCTAATCGGTTGGGATATCCTTGAAGATAAGCCCGATCTCTCCCAG
GAAGAGCTGGAGAGGATCAATCCATTTATATGGGAGGATGAATTTAAAGAGGTCTTCGCCAAAGGCGGTT
TTGATGCGGTAATTGGAAATCCGCCTTATATTAGAATTCAAATGATGAAGGAATGGGCTCCTGTAGAGGT
GGAATTTTACAAAGAGCATTACACGGTCGCCAAGAAAGGGAACTATGACGTTTATGTCGTATTCGTCGAA
AAGGGATTGGCCCTCCTGAACGAAAGCGGTCGTTTAGGTTTTATCCTACCAAATAAATTTTTTAATGCAC
AATATGGTTCACCGTTGCGTAGTTTATTATCAAATGGAAAAAATTTAGACGAAATTGTTAATTTTGGGCA
TGGACAAATATTCTGTGGCGTAACTACCTATACATGTCTGATCTTTCTGAATAAAATGCCAAAAGATTCA
TTCAAATATACATATGTCGAAGACTTGAATTCATGGAAAGAGGACGCATTATCAATAACGGGTGAAATTC
AAGCTAAGAATGCAGCATGTGCTGAATGGAATTTTATTGTTGGAAAAGGTTCAGATCTTTTTGATCGTTT
GAGTAAGATGCCTGTGAAGTTGGGAGATGTGGCTGAAAGGGTGTTTCAAGGGATCATTCCTGGAATGGAT
GCAGTTTATTCGATAAAATTGATCGGGGAAGATGATATTGTAATATGTTATTCGCGGGCTTTATCTAAAG
ATATTCAGATAGAAAGTAAAATTCTTCGTAAAATCGCCAGCGGTTCTCAGGTGAAGGCTTATACAATTGT
AGATGATAAATCAAGAGTTATCTATCCTTATCACTTTGAGGGAGATAATTGTGTTTTAATTCTGCCAGAT
AAGATGAAACAGGATTTTCCTTTGGCTTATGATTATCTTCAAAAAACCAGAGATCTATTGGACAAAAGAG
ATCGTGGCTCGGCTAAAGGAGCCCAATGGTATCGTTATATTAGAACCCAAAATATTGGATTACAAGCATA
TCCTAAGTTGGCCATCCCTCGCCTCGTCCATCGCTTGTGTGCAGCCTATGACGCAAATGCAGATTTTTGT
TTGGATAACGTGGATGTGGGTGGAGTGATTCTCTCTGAAAATAGCCCTGTTGGTTATATTTATATACTTG
GCTTATTAAATAGCAAGCTACTCAACTATTATTTTAAAATTAATAGTGTTCATTTTCGAGGTGGTTTTTT
CTCTGCTAATAGGCAATATATTGAACGTCTCCCCATTCGCACCATCGACTTCTCCGACCCCCAGGACGTC
ACCCGCCACGACAAGATGGTGAGCCTCGTGGAGACGATGCTCGACCTGCACAAACAACTCCAGGAAGTCG
GCACGCCACATGAAAAAACGCGCATCCAAAATCAGATCGGTTATACGGACAAGCAGATAGATGCCTTGGT
CTACGAACTGTACGACCTCACAGAGGAGGAGATCGCCATCGTGGAAGAGAGCACAAAATAG</span></span>
*GC% Content for gene: 7.886435%
*CDS Gene Sequence (codon optimized) - copy from output of Primer Design Protocol (paste as text only): N/a
*GC% Content for gene (codon optimized): N/a